BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Alpelisib | MK14 | 100.0 | 100 | nM |
Alpelisib | MK14 | 100.0 | 1000 | nM |
Alpelisib | MK11 | 100.0 | 100 | nM |
Alpelisib | MK11 | 97.0 | 1000 | nM |
Alpelisib | MK13 | 82.0 | 100 | nM |
Alpelisib | MK13 | 86.0 | 1000 | nM |
Alpelisib | MK12 | 80.0 | 100 | nM |
Alpelisib | MK12 | 90.0 | 1000 | nM |
Alpelisib | PAK1 | 75.0 | 100 | nM |
Alpelisib | PAK1 | 100.0 | 1000 | nM |
Alpelisib | PAK2 | 69.0 | 100 | nM |
Alpelisib | PAK2 | 89.0 | 1000 | nM |
Alpelisib | PAK3 | 96.0 | 100 | nM |
Alpelisib | PAK3 | 100.0 | 1000 | nM |
Alpelisib | PAK4 | 65.0 | 100 | nM |
Alpelisib | PAK4 | 91.0 | 1000 | nM |
Alpelisib | PAK6 | 89.0 | 100 | nM |
Alpelisib | PAK6 | 100.0 | 1000 | nM |
Alpelisib | PAK7 | 98.0 | 100 | nM |
Alpelisib | PAK7 | 97.0 | 1000 | nM |
Alpelisib | CDK16 | 100.0 | 100 | nM |
Alpelisib | CDK16 | 100.0 | 1000 | nM |
Alpelisib | PCTK2 | 100.0 | 100 | nM |
Alpelisib | PCTK2 | 100.0 | 1000 | nM |
Alpelisib | PCTK3 | 100.0 | 100 | nM |