BYL719 KINOMEscan - Dataset (ID:20263)

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Small Molecule Protein % Control Assay compound conc Conc unit
Alpelisib MK14 100.0 100
nM
Alpelisib MK14 100.0 1000
nM
Alpelisib MK11 100.0 100
nM
Alpelisib MK11 97.0 1000
nM
Alpelisib MK13 82.0 100
nM
Alpelisib MK13 86.0 1000
nM
Alpelisib MK12 80.0 100
nM
Alpelisib MK12 90.0 1000
nM
Alpelisib PAK1 75.0 100
nM
Alpelisib PAK1 100.0 1000
nM
Alpelisib PAK2 69.0 100
nM
Alpelisib PAK2 89.0 1000
nM
Alpelisib PAK3 96.0 100
nM
Alpelisib PAK3 100.0 1000
nM
Alpelisib PAK4 65.0 100
nM
Alpelisib PAK4 91.0 1000
nM
Alpelisib PAK6 89.0 100
nM
Alpelisib PAK6 100.0 1000
nM
Alpelisib PAK7 98.0 100
nM
Alpelisib PAK7 97.0 1000
nM
Alpelisib CDK16 100.0 100
nM
Alpelisib CDK16 100.0 1000
nM
Alpelisib PCTK2 100.0 100
nM
Alpelisib PCTK2 100.0 1000
nM
Alpelisib PCTK3 100.0 100
nM