Buparlisib KINOMEscan - Dataset (ID:20262)

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Small Molecule Protein % Control Assay compound conc Conc unit
Buparlisib PIK3CA(I800L) 0.0 100
nM
Buparlisib PIK3CA(I800L) 0.0 1000
nM
Buparlisib PIK3CA(E545K) 0.1 1000
nM
Buparlisib PIK3CA(E542K) 0.3 1000
nM
Buparlisib PIK3CA(C420R) 0.6 1000
nM
Buparlisib PIK3CA(E545A) 0.7 1000
nM
Buparlisib PIK3CA(Q546K) 0.7 1000
nM
Buparlisib PIK3CA(H1047L) 0.9 1000
nM
Buparlisib PIK3CA 1.4 1000
nM
Buparlisib MTOR 2.8 1000
nM
Buparlisib PIK3CA(H1047Y) 4.6 1000
nM
Buparlisib PIK3CA(M1043I) 4.7 1000
nM
Buparlisib PIK3CB 6.9 1000
nM
Buparlisib PIK3CA(E545K) 7.1 100
nM
Buparlisib PIK3CA(H1047Y) 12.0 100
nM
Buparlisib PIK3CA(C420R) 12.0 100
nM
Buparlisib PIK3CA(E545A) 12.0 100
nM
Buparlisib PIK3C3 14.0 1000
nM
Buparlisib PIK3CA(E542K) 15.0 100
nM
Buparlisib PIK3CA(M1043I) 15.0 100
nM
Buparlisib CSF1R-autoinhibited 21.0 1000
nM
Buparlisib PIK3CD 22.0 1000
nM
Buparlisib PIK3CA(Q546K) 23.0 100
nM
Buparlisib PIK3CA 27.0 100
nM
Buparlisib CLK4 28.0 1000
nM
  • Page 1 of 38
  • 1 to 25 of 936 records