Buparlisib KINOMEscan - Dataset (ID:20262)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Buparlisib | PIK3CA(I800L) | 0.0 | 100 | nM |
Buparlisib | PIK3CA(I800L) | 0.0 | 1000 | nM |
Buparlisib | PIK3CA(E545K) | 0.1 | 1000 | nM |
Buparlisib | PIK3CA(E542K) | 0.3 | 1000 | nM |
Buparlisib | PIK3CA(C420R) | 0.6 | 1000 | nM |
Buparlisib | PIK3CA(E545A) | 0.7 | 1000 | nM |
Buparlisib | PIK3CA(Q546K) | 0.7 | 1000 | nM |
Buparlisib | PIK3CA(H1047L) | 0.9 | 1000 | nM |
Buparlisib | PIK3CA | 1.4 | 1000 | nM |
Buparlisib | MTOR | 2.8 | 1000 | nM |
Buparlisib | PIK3CA(H1047Y) | 4.6 | 1000 | nM |
Buparlisib | PIK3CA(M1043I) | 4.7 | 1000 | nM |
Buparlisib | PIK3CB | 6.9 | 1000 | nM |
Buparlisib | PIK3CA(E545K) | 7.1 | 100 | nM |
Buparlisib | PIK3CA(H1047Y) | 12.0 | 100 | nM |
Buparlisib | PIK3CA(C420R) | 12.0 | 100 | nM |
Buparlisib | PIK3CA(E545A) | 12.0 | 100 | nM |
Buparlisib | PIK3C3 | 14.0 | 1000 | nM |
Buparlisib | PIK3CA(E542K) | 15.0 | 100 | nM |
Buparlisib | PIK3CA(M1043I) | 15.0 | 100 | nM |
Buparlisib | CSF1R-autoinhibited | 21.0 | 1000 | nM |
Buparlisib | PIK3CD | 22.0 | 1000 | nM |
Buparlisib | PIK3CA(Q546K) | 23.0 | 100 | nM |
Buparlisib | PIK3CA | 27.0 | 100 | nM |
Buparlisib | CLK4 | 28.0 | 1000 | nM |