GDC-0941 KINOMEscan-3 - Dataset (ID:20261)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Pictilisib | JNK3 | 93.0 | 1000 | nM |
| Pictilisib | KIT | 100.0 | 100 | nM |
| Pictilisib | KIT | 99.0 | 1000 | nM |
| Pictilisib | KIT(A829P) | 71.0 | 100 | nM |
| Pictilisib | KIT(A829P) | 100.0 | 1000 | nM |
| Pictilisib | KIT(D816H) | 88.0 | 100 | nM |
| Pictilisib | KIT(D816H) | 83.0 | 1000 | nM |
| Pictilisib | KIT(D816V) | 96.0 | 100 | nM |
| Pictilisib | KIT(D816V) | 97.0 | 1000 | nM |
| Pictilisib | KIT(L576P) | 100.0 | 100 | nM |
| Pictilisib | KIT(L576P) | 95.0 | 1000 | nM |
| Pictilisib | KIT(V559D) | 100.0 | 100 | nM |
| Pictilisib | KIT(V559D) | 100.0 | 1000 | nM |
| Pictilisib | KIT(V559D,T670I) | 100.0 | 100 | nM |
| Pictilisib | KIT(V559D,T670I) | 99.0 | 1000 | nM |
| Pictilisib | KIT(V559D,V654A) | 94.0 | 100 | nM |
| Pictilisib | KIT(V559D,V654A) | 100.0 | 1000 | nM |
| Pictilisib | KIT-autoinhibited | 72.0 | 100 | nM |
| Pictilisib | KIT-autoinhibited | 82.0 | 1000 | nM |
| Pictilisib | LATS1 | 100.0 | 100 | nM |
| Pictilisib | LATS1 | 100.0 | 1000 | nM |
| Pictilisib | LATS2 | 100.0 | 100 | nM |
| Pictilisib | LATS2 | 85.0 | 1000 | nM |
| Pictilisib | LCK | 82.0 | 100 | nM |
| Pictilisib | LCK | 85.0 | 1000 | nM |