Phosphorylation state and protein levels measured in BRAF(V600E/D) melanoma cell lines monitored by imaging - Dataset (ID:20219)
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Small Molecule | Cell Line | 2nd Drug | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Image | Measured Protein (Alexa Fluor 488) | Measured Protein Value (488) | Measured Protein (Alexa Fluor 568) | Measured Protein Value (568) | Measured Protein (Alexa Fluor 647) | Measured Protein Value (647) | Replicate | Plate Name | Plate Well |
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Vemurafenib | COLO 858 | 5.0000 | uM | 24 | hr | p27 Kip1 | 1100.60 | p-Rb(S807/S811) | 49.89 | p-ERK(T202/Y204) | 9.41 | 2 | Colo858-signal1 | C2 | ||
Vemurafenib | COLO 858 | 5.0000 | uM | 24 | hr | p27 Kip1 | 1101.80 | p-Rb(S807/S811) | 48.19 | p-ERK(T202/Y204) | 9.79 | 1 | Colo858-signal1 | B2 | ||
Vemurafenib | WM-115 | 5.0000 | uM | 24 | hr | p27 Kip1 | 333.60 | p-Rb(S807/S811) | 45.80 | p-ERK(T202/Y204) | 12.42 | 2 | WM115-signal1 | C2 | ||
Vemurafenib | WM-115 | 5.0000 | uM | 24 | hr | p27 Kip1 | 333.89 | p-Rb(S807/S811) | 50.05 | p-ERK(T202/Y204) | 12.54 | 1 | WM115-signal1 | B2 | ||
Vemurafenib | WM1552C | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 1000.20 | p-Rb(S807/S811) | 47.24 | p-cJun(S73) | 12.90 | 1 | WM1552C-signal3 | F3 | |
Vemurafenib | WM1552C | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 974.64 | p-Rb(S807/S811) | 46.90 | p-cJun(S73) | 13.63 | 2 | WM1552C-signal3 | G3 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.8000 | uM | 24 | hr | Ki-67 | 747.98 | p-Rb(S807/S811) | 47.12 | p-cJun(S73) | 13.64 | 2 | Colo858-signal3 | G4 | |
Vemurafenib | COLO 858 | 2.0000 | uM | 24 | hr | p27 Kip1 | 1016.50 | p-Rb(S807/S811) | 42.64 | p-ERK(T202/Y204) | 14.04 | 1 | Colo858-signal1 | B3 | ||
Vemurafenib | COLO 858 | 2.0000 | uM | 24 | hr | p27 Kip1 | 1027.10 | p-Rb(S807/S811) | 46.02 | p-ERK(T202/Y204) | 14.33 | 2 | Colo858-signal1 | C3 | ||
Vemurafenib | COLO 858 | 5.0000 | uM | 24 | hr | p-Histone H3(S10) | 265.46 | p-Rb(S807/S811) | 66.87 | p-S6(S235/S236 | 14.48 | 1 | Colo858-signal2 | B2 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 0.8000 | uM | 24 | hr | Ki-67 | 807.26 | p-Rb(S807/S811) | 48.49 | p-cJun(S73) | 14.54 | 1 | Colo858-signal3 | F4 | |
Vemurafenib | WM1552C | JNK-IN-8 | 5.0000 | uM | 24 | hr | Ki-67 | 1057.80 | p-Rb(S807/S811) | 58.43 | p-cJun(S73) | 14.63 | 1 | WM1552C-signal3 | F2 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 1130.80 | p-Rb(S807/S811) | 51.60 | p-cJun(S73) | 14.98 | 1 | Colo858-signal3 | F3 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 1116.10 | p-Rb(S807/S811) | 51.88 | p-cJun(S73) | 15.04 | 2 | Colo858-signal3 | G3 | |
Vemurafenib | WM-115 | 2.0000 | uM | 24 | hr | p27 Kip1 | 325.41 | p-Rb(S807/S811) | 43.62 | p-ERK(T202/Y204) | 15.11 | 1 | WM115-signal1 | B3 | ||
Vemurafenib | WM1552C | JNK-IN-8 | 5.0000 | uM | 24 | hr | Ki-67 | 1101.80 | p-Rb(S807/S811) | 60.49 | p-cJun(S73) | 15.34 | 2 | WM1552C-signal3 | G2 | |
Vemurafenib | WM-115 | 2.0000 | uM | 24 | hr | p27 Kip1 | 318.36 | p-Rb(S807/S811) | 43.44 | p-ERK(T202/Y204) | 16.10 | 2 | WM115-signal1 | C3 | ||
Vemurafenib | WM1552C | JNK-IN-8 | 5.0000 | uM | 24 | hr | p-Histone H3(S10) | 218.10 | p-Rb(S807/S811) | 64.53 | p-S6(S235/S236 | 16.11 | 1 | WM1552C-signal2 | F2 | |
Vemurafenib | COLO 858 | 5.0000 | uM | 24 | hr | p-Histone H3(S10) | 259.21 | p-Rb(S807/S811) | 68.62 | p-S6(S235/S236 | 16.39 | 2 | Colo858-signal2 | C2 | ||
Vemurafenib | COLO 858 | 0.8000 | uM | 24 | hr | p27 Kip1 | 1063.20 | p-Rb(S807/S811) | 48.29 | p-ERK(T202/Y204) | 17.48 | 1 | Colo858-signal1 | B4 | ||
Vemurafenib | WM-115 | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 657.65 | p-Rb(S807/S811) | 46.72 | p-cJun(S73) | 17.87 | 2 | WM115-signal3 | G3 | |
Vemurafenib | WM-115 | JNK-IN-8 | 2.0000 | uM | 24 | hr | Ki-67 | 684.33 | p-Rb(S807/S811) | 51.01 | p-cJun(S73) | 18.52 | 1 | WM115-signal3 | F3 | |
Vemurafenib | COLO 858 | 0.8000 | uM | 24 | hr | p27 Kip1 | 1014.60 | p-Rb(S807/S811) | 48.01 | p-ERK(T202/Y204) | 18.67 | 2 | Colo858-signal1 | C4 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 5.0000 | uM | 24 | hr | p-Histone H3(S10) | 416.80 | p-Rb(S807/S811) | 107.61 | p-S6(S235/S236 | 19.41 | 1 | Colo858-signal2 | F2 | |
Vemurafenib | LOXIMVI | JNK-IN-8 | 5.0000 | uM | 24 | hr | p-Histone H3(S10) | 358.85 | p-Rb(S807/S811) | 104.29 | p-S6(S235/S236 | 19.60 | 1 | LOXIMVI-signal2 | F2 |