Phosphorylation state and protein levels measured in BRAF(V600E/D) melanoma cell lines monitored by imaging - Dataset (ID:20219)
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Small Molecule | Cell Line | 2nd Drug | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Image | Measured Protein (Alexa Fluor 488) | Measured Protein Value (488) | Measured Protein (Alexa Fluor 568) | Measured Protein Value (568) | Measured Protein (Alexa Fluor 647) | Measured Protein Value (647) | Replicate | Plate Name | Plate Well |
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Vemurafenib | LOXIMVI | 0.0000 | uM | 24 | hr | p27 Kip1 | 346.49 | p-Rb(S807/S811) | 215.22 | p-ERK(T202/Y204) | 215.11 | 1 | LOXIMVI-signal1 | B11 | ||
Vemurafenib | LOXIMVI | JNK-IN-8 | 0.0000 | uM | 24 | hr | p27 Kip1 | 362.35 | p-Rb(S807/S811) | 212.69 | p-ERK(T202/Y204) | 226.97 | 1 | LOXIMVI-signal1 | F11 | |
Vemurafenib | COLO 858 | 0.0000 | uM | 24 | hr | Ki-67 | 2209.00 | p-Rb(S807/S811) | 151.07 | p-cJun(S73) | 28.62 | 1 | Colo858-signal3 | B11 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | Ki-67 | 2392.50 | p-Rb(S807/S811) | 158.97 | p-cJun(S73) | 29.83 | 2 | Colo858-signal3 | G11 | |
JNK-IN-8 | LOXIMVI | 0.0000 | uM | 24 | hr | p27 Kip1 | 348.21 | p-Rb(S807/S811) | 217.92 | p-ERK(T202/Y204) | 232.50 | 1 | LOXIMVI-signal1 | D11 | ||
JNK-IN-8 | LOXIMVI | 0.0000 | uM | 24 | hr | p27 Kip1 | 351.82 | p-Rb(S807/S811) | 222.97 | p-ERK(T202/Y204) | 225.84 | 2 | LOXIMVI-signal1 | E11 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 376.71 | p-Rb(S807/S811) | 165.48 | p-S6(S235/S236 | 397.13 | 2 | Colo858-signal2 | G11 | |
JNK-IN-8 | COLO 858 | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 357.02 | p-Rb(S807/S811) | 174.95 | p-S6(S235/S236 | 420.53 | 2 | Colo858-signal2 | E11 | ||
JNK-IN-8 | COLO 858 | 0.0000 | uM | 24 | hr | Ki-67 | 2186.70 | p-Rb(S807/S811) | 147.06 | p-cJun(S73) | 28.84 | 1 | Colo858-signal3 | D11 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | Ki-67 | 2257.00 | p-Rb(S807/S811) | 151.09 | p-cJun(S73) | 29.94 | 1 | Colo858-signal3 | F11 | |
Vemurafenib | LOXIMVI | 0.0000 | uM | 24 | hr | p27 Kip1 | 330.81 | p-Rb(S807/S811) | 208.35 | p-ERK(T202/Y204) | 212.82 | 2 | LOXIMVI-signal1 | C11 | ||
Vemurafenib | COLO 858 | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 358.86 | p-Rb(S807/S811) | 155.99 | p-S6(S235/S236 | 377.96 | 1 | Colo858-signal2 | B11 | ||
JNK-IN-8 | COLO 858 | 0.0000 | uM | 24 | hr | p27 Kip1 | 445.15 | p-Rb(S807/S811) | 158.36 | p-ERK(T202/Y204) | 601.12 | 2 | Colo858-signal1 | E11 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 336.86 | p-Rb(S807/S811) | 161.69 | p-S6(S235/S236 | 384.38 | 1 | Colo858-signal2 | F11 | |
Vemurafenib | COLO 858 | 0.0000 | uM | 24 | hr | p27 Kip1 | 479.59 | p-Rb(S807/S811) | 159.95 | p-ERK(T202/Y204) | 654.45 | 1 | Colo858-signal1 | B11 | ||
Vemurafenib | COLO 858 | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 377.25 | p-Rb(S807/S811) | 161.02 | p-S6(S235/S236 | 380.19 | 2 | Colo858-signal2 | C11 | ||
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | p27 Kip1 | 453.65 | p-Rb(S807/S811) | 157.18 | p-ERK(T202/Y204) | 608.40 | 1 | Colo858-signal1 | F11 | |
Vemurafenib | COLO 858 | JNK-IN-8 | 0.0000 | uM | 24 | hr | p27 Kip1 | 447.88 | p-Rb(S807/S811) | 161.30 | p-ERK(T202/Y204) | 568.39 | 2 | Colo858-signal1 | G11 | |
JNK-IN-8 | COLO 858 | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 323.83 | p-Rb(S807/S811) | 165.88 | p-S6(S235/S236 | 385.36 | 1 | Colo858-signal2 | D11 | ||
Vemurafenib | COLO 858 | 0.0000 | uM | 24 | hr | Ki-67 | 2259.80 | p-Rb(S807/S811) | 154.64 | p-cJun(S73) | 29.83 | 2 | Colo858-signal3 | C11 | ||
JNK-IN-8 | COLO 858 | 0.0000 | uM | 24 | hr | p27 Kip1 | 454.18 | p-Rb(S807/S811) | 159.65 | p-ERK(T202/Y204) | 628.56 | 1 | Colo858-signal1 | D11 | ||
JNK-IN-8 | COLO 858 | 0.0000 | uM | 24 | hr | Ki-67 | 2266.10 | p-Rb(S807/S811) | 152.55 | p-cJun(S73) | 28.74 | 2 | Colo858-signal3 | E11 | ||
Vemurafenib | COLO 858 | 0.0000 | uM | 24 | hr | p27 Kip1 | 452.92 | p-Rb(S807/S811) | 154.74 | p-ERK(T202/Y204) | 648.89 | 2 | Colo858-signal1 | C11 | ||
Vemurafenib | LOXIMVI | 0.0000 | uM | 24 | hr | p-Histone H3(S10) | 304.49 | p-Rb(S807/S811) | 234.76 | p-S6(S235/S236 | 449.34 | 1 | LOXIMVI-signal2 | B11 | ||
Vemurafenib | LOXIMVI | JNK-IN-8 | 0.0000 | uM | 24 | hr | p27 Kip1 | 351.99 | p-Rb(S807/S811) | 215.31 | p-ERK(T202/Y204) | 217.61 | 2 | LOXIMVI-signal1 | G11 |