GSK-461364A KINOMEscan - Dataset (ID:20194)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
GSK461364 | PLK1 | 0.1 | nM |
GSK461364 | SNARK | 23.0 | nM |
GSK461364 | LOK | 69.0 | nM |
GSK461364 | RSK2(Kin.Dom.1-N-terminal) | 190.0 | nM |
GSK461364 | PIM1 | 250.0 | nM |
GSK461364 | NEK2 | 260.0 | nM |
GSK461364 | RSK4(Kin.Dom.1-N-terminal) | 350.0 | nM |
GSK461364 | FLT3(D835H) | 410.0 | nM |
GSK461364 | FLT3(D835Y) | 430.0 | nM |
GSK461364 | BIKE | 470.0 | nM |
GSK461364 | PLK2 | 500.0 | nM |
GSK461364 | PKN2 | 620.0 | nM |
GSK461364 | FLT3 | 620.0 | nM |
GSK461364 | KCC2D | 620.0 | nM |
GSK461364 | FLT3(K663Q) | 650.0 | nM |
GSK461364 | FLT3(N841I) | 690.0 | nM |
GSK461364 | PLK3 | 740.0 | nM |
GSK461364 | RPS6KA4(Kin.Dom.2-C-terminal) | 740.0 | nM |
GSK461364 | PIP5K1A | 770.0 | nM |
GSK461364 | CSNK2A2 | 990.0 | nM |
GSK461364 | CAMK2A | 1000.0 | nM |
GSK461364 | SLK | 1100.0 | nM |
GSK461364 | PIM3 | 1100.0 | nM |
GSK461364 | NEK9 | 1100.0 | nM |
GSK461364 | NEK5 | 1100.0 | nM |