PKC-412 KINOMEscan - Dataset (ID:20187)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| PKC412 | FLT3(K663Q) | 2.0 | nM |
| PKC412 | FLT3(N841I) | 6.0 | nM |
| PKC412 | FLT3(D835H) | 6.8 | nM |
| PKC412 | KIT(D816V) | 7.7 | nM |
| PKC412 | EGFR(L858R,T790M) | 8.8 | nM |
| PKC412 | TBK1 | 9.3 | nM |
| PKC412 | PKN1 | 9.3 | nM |
| PKC412 | EGFR(T790M) | 9.8 | nM |
| PKC412 | FLT3(ITD) | 11.0 | nM |
| PKC412 | FLT3 | 11.0 | nM |
| PKC412 | JAK3(JH1domain-catalytic) | 12.0 | nM |
| PKC412 | FLT3(R834Q) | 12.0 | nM |
| PKC412 | PKN2 | 15.0 | nM |
| PKC412 | YSK4 | 15.0 | nM |
| PKC412 | FLT3(D835Y) | 15.0 | nM |
| PKC412 | MLK1 | 15.0 | nM |
| PKC412 | KIT(D816H) | 16.0 | nM |
| PKC412 | MLK3 | 17.0 | nM |
| PKC412 | RET(V804M) | 20.0 | nM |
| PKC412 | CAMK2A | 20.0 | nM |
| PKC412 | MARK3 | 21.0 | nM |
| PKC412 | RET(V804L) | 27.0 | nM |
| PKC412 | KCC2D | 36.0 | nM |
| PKC412 | GCN2(Kin.Dom.2,S808G) | 39.0 | nM |
| PKC412 | MST1 | 40.0 | nM |