KW-2449 KINOMEscan - Dataset (ID:20185)

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Small Molecule Protein Kd Conc unit
KW2449 DRAK1 2.9
nM
KW2449 MLCK 4.3
nM
KW2449 DRAK2 4.8
nM
KW2449 YSK4 5.2
nM
KW2449 ABL1(T315I)-phosphorylated 5.9
nM
KW2449 FLT3(K663Q) 6.6
nM
KW2449 BIKE 9.6
nM
KW2449 MAP4K2 11.0
nM
KW2449 ABL1(T315I)-nonphosphorylated 12.0
nM
KW2449 KIT(V559D,T670I) 12.0
nM
KW2449 FLT3(N841I) 13.0
nM
KW2449 FLT3(D835Y) 13.0
nM
KW2449 SLK 13.0
nM
KW2449 FLT3(D835H) 13.0
nM
KW2449 LOK 13.0
nM
KW2449 SRPK2 15.0
nM
KW2449 FLT3 15.0
nM
KW2449 ABL1(H396P)-nonphosphorylated 17.0
nM
KW2449 YES 18.0
nM
KW2449 ABL1(M351T)-phosphorylated 19.0
nM
KW2449 FLT3(ITD) 20.0
nM
KW2449 PLK4 21.0
nM
KW2449 KIT(L576P) 21.0
nM
KW2449 ABL1(Q252H)-phosphorylated 22.0
nM
KW2449 KIT(V559D) 23.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records