KW-2449 KINOMEscan - Dataset (ID:20185)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
KW2449 | DRAK1 | 2.9 | nM |
KW2449 | MLCK | 4.3 | nM |
KW2449 | DRAK2 | 4.8 | nM |
KW2449 | YSK4 | 5.2 | nM |
KW2449 | ABL1(T315I)-phosphorylated | 5.9 | nM |
KW2449 | FLT3(K663Q) | 6.6 | nM |
KW2449 | BIKE | 9.6 | nM |
KW2449 | MAP4K2 | 11.0 | nM |
KW2449 | ABL1(T315I)-nonphosphorylated | 12.0 | nM |
KW2449 | KIT(V559D,T670I) | 12.0 | nM |
KW2449 | FLT3(N841I) | 13.0 | nM |
KW2449 | FLT3(D835Y) | 13.0 | nM |
KW2449 | SLK | 13.0 | nM |
KW2449 | FLT3(D835H) | 13.0 | nM |
KW2449 | LOK | 13.0 | nM |
KW2449 | SRPK2 | 15.0 | nM |
KW2449 | FLT3 | 15.0 | nM |
KW2449 | ABL1(H396P)-nonphosphorylated | 17.0 | nM |
KW2449 | YES | 18.0 | nM |
KW2449 | ABL1(M351T)-phosphorylated | 19.0 | nM |
KW2449 | FLT3(ITD) | 20.0 | nM |
KW2449 | PLK4 | 21.0 | nM |
KW2449 | KIT(L576P) | 21.0 | nM |
KW2449 | ABL1(Q252H)-phosphorylated | 22.0 | nM |
KW2449 | KIT(V559D) | 23.0 | nM |