ABT-869 KINOMEscan - Dataset (ID:20182)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Linifanib | FLT3 | 0.6 | nM |
| Linifanib | FLT3(K663Q) | 1.3 | nM |
| Linifanib | KIT(V559D) | 1.7 | nM |
| Linifanib | KIT(L576P) | 1.9 | nM |
| Linifanib | PGFRB | 1.9 | nM |
| Linifanib | KIT | 2.0 | nM |
| Linifanib | FLT3(N841I) | 2.6 | nM |
| Linifanib | FLT3(D835H) | 2.7 | nM |
| Linifanib | CSF1R | 3.4 | nM |
| Linifanib | KIT(V559D,T670I) | 3.8 | nM |
| Linifanib | PGFRA | 4.2 | nM |
| Linifanib | VGFR1 | 7.5 | nM |
| Linifanib | VGFR2 | 8.1 | nM |
| Linifanib | FLT3(ITD) | 8.8 | nM |
| Linifanib | MUSK | 10.0 | nM |
| Linifanib | FLT3(D835Y) | 11.0 | nM |
| Linifanib | FLT4 | 16.0 | nM |
| Linifanib | FLT3(R834Q) | 16.0 | nM |
| Linifanib | KIT(A829P) | 17.0 | nM |
| Linifanib | KIT(V559D,V654A) | 21.0 | nM |
| Linifanib | EPHB6 | 33.0 | nM |
| Linifanib | CDC2L5 | 38.0 | nM |
| Linifanib | HIPK4 | 46.0 | nM |
| Linifanib | RET(V804M) | 54.0 | nM |
| Linifanib | DDR1 | 58.0 | nM |