GSK-1363089 KINOMEscan - Dataset (ID:20176)

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Small Molecule Protein Kd Conc unit
Foretinib AXL 0.1
nM
Foretinib DDR1 0.2
nM
Foretinib MERTK 0.3
nM
Foretinib LOK 0.5
nM
Foretinib HIPK4 0.5
nM
Foretinib RET(M918T) 0.7
nM
Foretinib RET 0.7
nM
Foretinib FLT3(K663Q) 0.8
nM
Foretinib TIE1 0.8
nM
Foretinib MET(Y1235D) 0.8
nM
Foretinib FLT3 0.9
nM
Foretinib EPHA3 1.0
nM
Foretinib PGFRB 1.0
nM
Foretinib MET(M1250T) 1.0
nM
Foretinib EPHA6 1.1
nM
Foretinib EPHB6 1.3
nM
Foretinib FLT3(D835H) 1.4
nM
Foretinib MET 1.4
nM
Foretinib FLT3(N841I) 1.5
nM
Foretinib FLT4 1.5
nM
Foretinib RET(V804L) 1.6
nM
Foretinib CSF1R 1.8
nM
Foretinib EPHA8 1.8
nM
Foretinib EPHA4 1.9
nM
Foretinib FLT3(D835Y) 2.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records