GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Foretinib | AXL | 0.1 | nM |
Foretinib | DDR1 | 0.2 | nM |
Foretinib | MERTK | 0.3 | nM |
Foretinib | LOK | 0.5 | nM |
Foretinib | HIPK4 | 0.5 | nM |
Foretinib | RET(M918T) | 0.7 | nM |
Foretinib | RET | 0.7 | nM |
Foretinib | FLT3(K663Q) | 0.8 | nM |
Foretinib | TIE1 | 0.8 | nM |
Foretinib | MET(Y1235D) | 0.8 | nM |
Foretinib | FLT3 | 0.9 | nM |
Foretinib | EPHA3 | 1.0 | nM |
Foretinib | PGFRB | 1.0 | nM |
Foretinib | MET(M1250T) | 1.0 | nM |
Foretinib | EPHA6 | 1.1 | nM |
Foretinib | EPHB6 | 1.3 | nM |
Foretinib | FLT3(D835H) | 1.4 | nM |
Foretinib | MET | 1.4 | nM |
Foretinib | FLT3(N841I) | 1.5 | nM |
Foretinib | FLT4 | 1.5 | nM |
Foretinib | RET(V804L) | 1.6 | nM |
Foretinib | CSF1R | 1.8 | nM |
Foretinib | EPHA8 | 1.8 | nM |
Foretinib | EPHA4 | 1.9 | nM |
Foretinib | FLT3(D835Y) | 2.0 | nM |