BIBF-1120 KINOMEscan - Dataset (ID:20175)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Nintedanib | FLT3(D835Y) | 0.4 | nM |
| Nintedanib | FLT3(D835H) | 0.7 | nM |
| Nintedanib | FLT3(ITD) | 0.7 | nM |
| Nintedanib | MP2K5 | 1.8 | nM |
| Nintedanib | BIKE | 2.2 | nM |
| Nintedanib | FLT3(N841I) | 2.6 | nM |
| Nintedanib | KIT(L576P) | 2.7 | nM |
| Nintedanib | VGFR2 | 2.9 | nM |
| Nintedanib | KIT(V559D,T670I) | 2.9 | nM |
| Nintedanib | PKNB(M.tuberculosis) | 3.6 | nM |
| Nintedanib | FLT3 | 3.8 | nM |
| Nintedanib | TAK1 | 4.1 | nM |
| Nintedanib | TRKA | 4.5 | nM |
| Nintedanib | FLT3(K663Q) | 4.5 | nM |
| Nintedanib | JAK1(JH2domain-pseudokinase) | 4.8 | nM |
| Nintedanib | MELK | 4.9 | nM |
| Nintedanib | YSK4 | 5.2 | nM |
| Nintedanib | KIT | 5.7 | nM |
| Nintedanib | LCK | 6.2 | nM |
| Nintedanib | KIT(V559D) | 6.3 | nM |
| Nintedanib | JAK3(JH1domain-catalytic) | 8.2 | nM |
| Nintedanib | PRP4 | 8.4 | nM |
| Nintedanib | MERTK | 8.5 | nM |
| Nintedanib | CLK1 | 8.8 | nM |
| Nintedanib | MST1 | 9.0 | nM |