Erlotinib KINOMEscan - Dataset (ID:20160)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Erlotinib | EGFR(L747-T751del,Sins) | 0.4 | nM |
Erlotinib | EGFR(G719S) | 0.5 | nM |
Erlotinib | EGFR(L747-S752del, P753S) | 0.5 | nM |
Erlotinib | EGFR(L747-E749del, A750P) | 0.5 | nM |
Erlotinib | EGFR(E746-A750del) | 0.5 | nM |
Erlotinib | EGFR | 0.7 | nM |
Erlotinib | EGFR(G719C) | 0.9 | nM |
Erlotinib | EGFR(L858R) | 1.0 | nM |
Erlotinib | EGFR(L861Q) | 1.2 | nM |
Erlotinib | EGFR(S752-I759del) | 1.6 | nM |
Erlotinib | GAK | 3.1 | nM |
Erlotinib | LOK | 19.0 | nM |
Erlotinib | YSK4 | 25.0 | nM |
Erlotinib | SLK | 26.0 | nM |
Erlotinib | ABL1(H396P)-phosphorylated | 58.0 | nM |
Erlotinib | ABL1(T315I)-phosphorylated | 59.0 | nM |
Erlotinib | ABL1(Q252H)-phosphorylated | 61.0 | nM |
Erlotinib | ABL1(E255K)-phosphorylated | 63.0 | nM |
Erlotinib | ABL1(M351T)-phosphorylated | 66.0 | nM |
Erlotinib | ABL1(Y253F)-phosphorylated | 76.0 | nM |
Erlotinib | ABL1-phosphorylated | 76.0 | nM |
Erlotinib | ABL1(H396P)-nonphosphorylated | 89.0 | nM |
Erlotinib | MP2K5 | 96.0 | nM |
Erlotinib | FLT3(D835Y) | 130.0 | nM |
Erlotinib | EGFR(T790M) | 140.0 | nM |