AMG-706 KINOMEscan - Dataset (ID:20150)

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Small Molecule Protein Kd Conc unit
Motesanib KIT(L576P) 1.3
nM
Motesanib KIT(V559D) 3.2
nM
Motesanib KIT 3.7
nM
Motesanib CSF1R 5.6
nM
Motesanib MLTK 8.0
nM
Motesanib PGFRB 9.1
nM
Motesanib FLT4 9.7
nM
Motesanib PGFRA 10.0
nM
Motesanib VGFR1 12.0
nM
Motesanib KIT(V559D,T670I) 13.0
nM
Motesanib RET 14.0
nM
Motesanib KIT(A829P) 15.0
nM
Motesanib RET(M918T) 20.0
nM
Motesanib KIT(V559D,V654A) 23.0
nM
Motesanib VGFR2 26.0
nM
Motesanib FLT3(K663Q) 54.0
nM
Motesanib FLT3 71.0
nM
Motesanib FRK 99.0
nM
Motesanib LYN 160.0
nM
Motesanib KIT(D816H) 180.0
nM
Motesanib YSK4 200.0
nM
Motesanib TNNI3K 220.0
nM
Motesanib DDR1 260.0
nM
Motesanib BRAF(V600E) 280.0
nM
Motesanib CIT 300.0
nM
  • Page 1 of 18
  • 1 to 25 of 442 records