BI-2536 KINOMEscan-2 - Dataset (ID:20149)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
BI-2536 | PLK1 | 0.2 | nM |
BI-2536 | PLK2 | 0.8 | nM |
BI-2536 | PLK3 | 4.0 | nM |
BI-2536 | RPS6KA4(Kin.Dom.2-C-terminal) | 12.0 | nM |
BI-2536 | KKCC1 | 22.0 | nM |
BI-2536 | CAMKK2 | 23.0 | nM |
BI-2536 | MYLK | 97.0 | nM |
BI-2536 | PI42C | 110.0 | nM |
BI-2536 | DAPK3 | 130.0 | nM |
BI-2536 | FAK1 | 150.0 | nM |
BI-2536 | ALK | 160.0 | nM |
BI-2536 | GAK | 180.0 | nM |
BI-2536 | EGFR(L858R,T790M) | 240.0 | nM |
BI-2536 | RPS6KA5(Kin.Dom.2-C-terminal) | 270.0 | nM |
BI-2536 | FAK2 | 310.0 | nM |
BI-2536 | KPCD1 | 320.0 | nM |
BI-2536 | KPCD3 | 350.0 | nM |
BI-2536 | EGFR(T790M) | 360.0 | nM |
BI-2536 | CSNK1E | 380.0 | nM |
BI-2536 | CLK2 | 460.0 | nM |
BI-2536 | PRKR | 460.0 | nM |
BI-2536 | YSK4 | 480.0 | nM |
BI-2536 | KPCD2 | 510.0 | nM |
BI-2536 | DAPK1 | 540.0 | nM |
BI-2536 | CLK3 | 630.0 | nM |