R406 KINOMEscan-2 - Dataset (ID:20148)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
R406 | FLT3(D835Y) | 0.4 | nM |
R406 | FLT3(ITD) | 0.5 | nM |
R406 | FLT3 | 0.7 | nM |
R406 | FLT3(K663Q) | 0.7 | nM |
R406 | FLT3(D835H) | 0.7 | nM |
R406 | FLT3(N841I) | 1.5 | nM |
R406 | STK16 | 1.7 | nM |
R406 | RET(V804L) | 2.2 | nM |
R406 | KIT(D816V) | 2.5 | nM |
R406 | RET(V804M) | 3.1 | nM |
R406 | PGFRB | 3.3 | nM |
R406 | GCN2(Kin.Dom.2,S808G) | 3.3 | nM |
R406 | KIT(A829P) | 3.5 | nM |
R406 | JAK2(JH1domain-catalytic) | 3.5 | nM |
R406 | MLK2 | 3.8 | nM |
R406 | RET(M918T) | 4.1 | nM |
R406 | RET | 4.1 | nM |
R406 | PLK4 | 4.2 | nM |
R406 | MLK1 | 4.3 | nM |
R406 | FLT3(R834Q) | 4.4 | nM |
R406 | PLK3 | 5.1 | nM |
R406 | KIT(L576P) | 5.6 | nM |
R406 | KIT(V559D) | 5.7 | nM |
R406 | NEK6 | 6.3 | nM |
R406 | KIT(D816H) | 6.5 | nM |