R406 KINOMEscan-2 - Dataset (ID:20148)

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Small Molecule Protein Kd Conc unit
R406 FLT3(D835Y) 0.4
nM
R406 FLT3(ITD) 0.5
nM
R406 FLT3 0.7
nM
R406 FLT3(K663Q) 0.7
nM
R406 FLT3(D835H) 0.7
nM
R406 FLT3(N841I) 1.5
nM
R406 STK16 1.7
nM
R406 RET(V804L) 2.2
nM
R406 KIT(D816V) 2.5
nM
R406 RET(V804M) 3.1
nM
R406 PGFRB 3.3
nM
R406 GCN2(Kin.Dom.2,S808G) 3.3
nM
R406 KIT(A829P) 3.5
nM
R406 JAK2(JH1domain-catalytic) 3.5
nM
R406 MLK2 3.8
nM
R406 RET(M918T) 4.1
nM
R406 RET 4.1
nM
R406 PLK4 4.2
nM
R406 MLK1 4.3
nM
R406 FLT3(R834Q) 4.4
nM
R406 PLK3 5.1
nM
R406 KIT(L576P) 5.6
nM
R406 KIT(V559D) 5.7
nM
R406 NEK6 6.3
nM
R406 KIT(D816H) 6.5
nM
  • Page 1 of 18
  • 1 to 25 of 442 records