AZD4547 KINOMEscan - Dataset (ID:20129)

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Small Molecule Protein % Control Assay compound conc Conc unit
AZD4547 AAK1 14.0 10
uM
AZD4547 ABL1(E255K)-phosphorylated 2.0 10
uM
AZD4547 ABL1(F317I)-nonphosphorylated 64.0 10
uM
AZD4547 ABL1(F317I)-phosphorylated 25.0 10
uM
AZD4547 ABL1(F317L)-nonphosphorylated 19.0 10
uM
AZD4547 ABL1(F317L)-phosphorylated 8.2 10
uM
AZD4547 ABL1(H396P)-nonphosphorylated 0.1 10
uM
AZD4547 ABL1(H396P)-phosphorylated 2.3 10
uM
AZD4547 ABL1(M351T)-phosphorylated 2.3 10
uM
AZD4547 ABL1-nonphosphorylated 1.4 10
uM
AZD4547 ABL1-phosphorylated 2.6 10
uM
AZD4547 ABL1(Q252H)-nonphosphorylated 1.4 10
uM
AZD4547 ABL1(Q252H)-phosphorylated 2.0 10
uM
AZD4547 ABL1(T315I)-nonphosphorylated 0.0 10
uM
AZD4547 ABL1(T315I)-phosphorylated 0.3 10
uM
AZD4547 ABL1(Y253F)-phosphorylated 0.9 10
uM
AZD4547 ABL2 13.0 10
uM
AZD4547 ACVR1 41.0 10
uM
AZD4547 ACVR1B 88.0 10
uM
AZD4547 ACVR2A 100.0 10
uM
AZD4547 ACVR2B 70.0 10
uM
AZD4547 ACVRL1 100.0 10
uM
AZD4547 ADCK3 95.0 10
uM
AZD4547 ADCK4 100.0 10
uM
AZD4547 AKT1 100.0 10
uM
  • Page 1 of 19
  • 1 to 25 of 456 records