BS-181 KINOMEscan - Dataset (ID:20127)

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Small Molecule Protein % Control Assay compound conc Conc unit
BS-181 ABL1(E255K)-phosphorylated 70.0 10
uM
BS-181 ABL1(F317I)-nonphosphorylated 88.0 10
uM
BS-181 ABL1(F317I)-phosphorylated 77.0 10
uM
BS-181 ABL1(F317L)-nonphosphorylated 96.0 10
uM
BS-181 ABL1(F317L)-phosphorylated 87.0 10
uM
BS-181 ABL1(H396P)-nonphosphorylated 93.0 10
uM
BS-181 ABL1(H396P)-phosphorylated 88.0 10
uM
BS-181 ABL1(M351T)-phosphorylated 100.0 10
uM
BS-181 ABL1(Q252H)-nonphosphorylated 100.0 10
uM
BS-181 ABL1(Q252H)-phosphorylated 89.0 10
uM
BS-181 ABL1(T315I)-nonphosphorylated 93.0 10
uM
BS-181 ABL1(T315I)-phosphorylated 88.0 10
uM
BS-181 ABL1(Y253F)-phosphorylated 78.0 10
uM
BS-181 ABL1-nonphosphorylated 96.0 10
uM
BS-181 ABL1-phosphorylated 84.0 10
uM
BS-181 ABL2 90.0 10
uM
BS-181 ACVR1 100.0 10
uM
BS-181 ACVR1B 100.0 10
uM
BS-181 ACVR2A 92.0 10
uM
BS-181 ACVR2B 83.0 10
uM
BS-181 ACVRL1 75.0 10
uM
BS-181 ADCK3 100.0 10
uM
BS-181 ADCK4 86.0 10
uM
BS-181 AKT1 100.0 10
uM
BS-181 AAK1 100.0 10
uM
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