Metrics other than potency reveal systematic variation in responses to cancer drugs - Dataset (ID:20120)

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Small Molecule Cell Line log10[max. dose (M)] R^2 (goodness of fit) log10[EC50 (M)] log10[IC50 (M)] log10[GI50 (M)] HillSlope E_inf E_max AUC
Tozasertib HCC38 -4.0000 0.9362 -6.0550 -6.0552 -6.5583 0.5106 0.0000 0.0819 5.5362
Tozasertib HCC70 -4.0000 0.7843 -5.2470 -5.2466 NaN 0.3821 0.0000 0.2503 6.3077
Tozasertib HCC1419 -4.0000 0.8498 -4.1981 -4.1981 -4.8568 0.9298 0.0000 0.3956 7.7843
Tozasertib HCC1569 -4.0000 0.9023 -5.0220 -5.0220 -5.7245 0.5522 0.0000 0.2143 6.7476
Tozasertib BT-549 -4.0000 0.9135 -5.5800 -5.5799 -5.7199 0.6894 0.0000 0.0753 6.3599
Tozasertib MDA-MB-231 -4.0000 0.9221 -4.8628 -4.8630 -4.9264 1.1070 0.0000 0.0998 7.3371
Tozasertib HCC1395 -4.0000 0.9267 -4.9570 -4.9570 -5.7943 0.9915 0.0000 0.1011 6.6654
GSK461364 MDA-MB-175-VII -4.4776 0.7103 -4.6478 -4.6477 -4.9999 1.7670 0.0000 0.3335 7.1799
GSK461364 MCF12A -4.4776 0.7888 -5.5836 -5.5839 -5.8310 0.4970 0.0000 0.2199 6.8984
GSK461364 UACC-812 -4.4776 0.8943 -4.8642 -4.8641 -5.0359 3.7120 0.0000 0.0354 8.8806
Tozasertib BT-474 -4.0000 0.8143 -4.4178 -4.4177 -5.1819 1.5550 0.0000 0.1831 7.9621
GSK461364 600MPE -4.4776 0.8618 -4.8362 -4.8362 -4.8631 4.0000 0.0000 0.0355 7.9370
GSK461364 HCC1569 -4.4776 0.7965 -5.0714 -5.0714 -5.7745 0.3696 0.0000 0.3763 6.5207
GSK461364 BT-483 -4.4776 0.8228 -4.9223 -4.9223 -5.7449 2.2735 0.0000 0.0889 7.5231
Tozasertib BT-20 -4.0000 0.8366 -4.6124 -4.6124 -5.5324 0.4999 0.0000 0.3307 7.0328
GSK461364 LY2 -4.4776 0.7525 -5.3501 -5.3501 -5.9259 0.3841 0.0000 0.3161 6.7154
GSK461364 MCF 10F -4.4776 0.8285 -6.0156 -6.0160 -7.2051 0.4255 0.0000 0.2392 6.1498
GSK461364 HCC1428 -4.4776 0.9592 -4.9400 -4.9399 -5.2690 3.3400 0.0000 0.0203 7.7381
GSK461364 184B5 -4.4776 0.7303 -5.5881 -5.5882 -6.3658 0.4307 0.0000 0.2496 6.7499
GSK461364 T47D -4.4776 0.7866 -4.9834 -4.9834 -6.1129 1.8790 0.0000 0.1008 7.2108
GSK461364 SUM185PE -4.4776 0.8273 -5.1574 -5.1573 -5.8411 1.7260 0.0000 0.0879 7.3788
GSK461364 184A1 -4.4776 0.9640 -4.8844 -4.8844 -5.2355 2.3020 0.0000 0.1037 7.8611
GSK461364 BT-474 -4.4776 0.7677 -4.9305 -4.9304 -5.0842 3.9990 0.0000 0.0152 7.4055
Tozasertib MDA-MB-157 -4.0000 0.9065 -5.0270 -5.0273 -5.4475 0.8482 0.0000 0.1185 6.9191
Tozasertib MDA-MB-134-VI -4.0000 0.9695 -4.7252 -4.7252 -5.7263 0.4520 0.0000 0.3198 7.0698
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