XMD-12 KINOMEscan - Dataset (ID:20115)
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| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| XMD-12 | ABL1(H396P)-nonphosphorylated | 0.2 | 1 | uM |
| XMD-12 | M3K2 | 0.2 | 1 | uM |
| XMD-12 | ERK5 | 0.3 | 1 | uM |
| XMD-12 | ABL1(Q252H)-phosphorylated | 0.4 | 1 | uM |
| XMD-12 | MAP3K3 | 0.4 | 1 | uM |
| XMD-12 | TAOK2 | 0.6 | 1 | uM |
| XMD-12 | DCAMKL2 | 0.6 | 1 | uM |
| XMD-12 | ABL1(E255K)-phosphorylated | 0.6 | 1 | uM |
| XMD-12 | TAOK1 | 0.9 | 1 | uM |
| XMD-12 | LRRK2(G2019S) | 0.9 | 1 | uM |
| XMD-12 | TNK1 | 1.0 | 1 | uM |
| XMD-12 | ABL1(T315I)-phosphorylated | 1.0 | 1 | uM |
| XMD-12 | TAOK3 | 1.2 | 1 | uM |
| XMD-12 | JAK2(JH1domain-catalytic) | 1.3 | 1 | uM |
| XMD-12 | AURKB | 1.4 | 1 | uM |
| XMD-12 | RET(V804L) | 1.7 | 1 | uM |
| XMD-12 | DCLK1 | 1.8 | 1 | uM |
| XMD-12 | PLK4 | 1.8 | 1 | uM |
| XMD-12 | TYK2(JH1domain-catalytic) | 1.9 | 1 | uM |
| XMD-12 | ABL1(Y253F)-phosphorylated | 1.9 | 1 | uM |
| XMD-12 | ABL1(Q252H)-nonphosphorylated | 2.1 | 1 | uM |
| XMD-12 | LRRK2 | 2.2 | 1 | uM |
| XMD-12 | AURKA | 2.4 | 1 | uM |
| XMD-12 | ABL1(H396P)-phosphorylated | 2.4 | 1 | uM |
| XMD-12 | RET(V804M) | 3.0 | 1 | uM |