AG1478 KINOMEscan - Dataset (ID:20086)

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Small Molecule Protein % Control Assay compound conc Conc unit
AG1478 ABL1(E255K)-phosphorylated 6.6 10
uM
AG1478 ABL1(F317I)-nonphosphorylated 18.0 10
uM
AG1478 ABL1(F317I)-phosphorylated 26.0 10
uM
AG1478 ABL1(F317L)-nonphosphorylated 6.8 10
uM
AG1478 ABL1(F317L)-phosphorylated 9.2 10
uM
AG1478 ABL1(H396P)-nonphosphorylated 2.2 10
uM
AG1478 ABL1(H396P)-phosphorylated 0.7 10
uM
AG1478 ABL1(M351T)-phosphorylated 1.4 10
uM
AG1478 ABL1(Q252H)-nonphosphorylated 6.7 10
uM
AG1478 ABL1(Q252H)-phosphorylated 7.1 10
uM
AG1478 ABL1(T315I)-nonphosphorylated 12.0 10
uM
AG1478 ABL1(T315I)-phosphorylated 2.5 10
uM
AG1478 ABL1(Y253F)-phosphorylated 2.3 10
uM
AG1478 ABL1-nonphosphorylated 3.4 10
uM
AG1478 ABL1-phosphorylated 0.9 10
uM
AG1478 ABL2 34.0 10
uM
AG1478 ACVR1 74.0 10
uM
AG1478 ACVR1B 100.0 10
uM
AG1478 ACVR2A 92.0 10
uM
AG1478 ACVR2B 54.0 10
uM
AG1478 ACVRL1 100.0 10
uM
AG1478 ADCK3 56.0 10
uM
AG1478 ADCK4 28.0 10
uM
AG1478 AKT1 100.0 10
uM
AG1478 AAK1 18.0 10
uM
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