Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 2 of 2: Calculated dose response metrics - Dataset (ID:20344)

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Cell Small Molecule Primary Target Pathway GR50 GRmax GR_AOC Death_AUC GR Hill Coefficient GEC50 GR r2
MDA-MB-134-VI Cediranib
VEGFR/cKIT
RTK
4.2103
-0.9999 0.0977 0.0979 5.0000
5.2449
0.99321
MDA-MB-134-VI Ceritinib
ALK
RTK
0.13159
-0.9992 0.6654 0.1723 0.9173
0.43587
0.98922
MDA-MB-134-VI Abemaciclib
CDK4/6
Cell cycle
Inf
-0.9986 0.5722 0.0709 0.0000
Inf
0.086291
MDA-MB-361 Ceritinib
ALK
RTK
0.26636
-0.9910 0.5462 0.1443 0.8263
1.0067
0.97236
MDA-MB-361 Taselisib
PI3Ka, g, d
PI3K/mTOR
0.0017737
-0.9902 1.4103 0.4329 0.6207
0.010237
0.9975
MDA-MB-361 Cediranib
VEGFR/cKIT
RTK
2.2171
-0.9803 0.2895 0.1040 2.2939
3.5791
0.96048
MDA-MB-361 Torin2
mTOR/ATM/ATR
PI3K/mTOR
0.0050713
-0.9642 0.8689 0.2561 0.9911
0.014575
0.99687
MDA-MB-361 Buparlisib
pan PI3K
PI3K/mTOR
0.21797
-0.9584 0.6114 0.1763 0.9709
0.67584
0.99384
HCC1500 Ceritinib
ALK
RTK
1.4068
-0.9535 0.2988 0.1206 1.5745
2.8266
0.97255
MDA-MB-134-VI Torin2
mTOR/ATM/ATR
PI3K/mTOR
0.0051713
-0.9461 0.8935 0.2182 1.1423
0.01301
0.99597
MDA-MB-134-VI Doxorubicin
Chemo
Chemotherapy
0.0033105
-0.9458 1.1481 0.2491 0.9132
0.010163
0.97259
PDX1328 Ceritinib
ALK
RTK
0.25503
-0.9426 0.5536 0.1190 0.8974
0.86749
0.9878
MDA-MB-361 Vorinostat
HDAC
Misc
0.76224
-0.9392 0.4607 0.1761 2.2187
1.2401
0.99784
MDA-MB-361 Pictilisib
pan PI3K
PI3K/mTOR
0.079201
-0.9375 0.7161 0.1619 0.6291
0.45409
0.98391
MDA-MB-157 Ceritinib
ALK
RTK
0.48405
-0.9264 0.4600 0.1138 0.9467
1.5449
0.97503
PDX1328 Topotecan
Topo I
Chemotherapy
0.0059222
-0.9128 1.0720 0.1509 0.4616
0.063175
0.94441
MDA-MB-157 Dinaciclib
pan CDK
Cell cycle
0.017724
-0.9106 0.7675 0.3195 3.8857
0.023072
0.99901
HCC70 Dinaciclib
pan CDK
Cell cycle
0.01286
-0.9093 0.8338 0.3254 5.0000
0.015807
0.9991
PDX1328 ABT-737
Bcl2/XL
Misc
1.0279
-0.8967 0.3548 0.1542 1.3255
2.3546
0.97784
MDA-MB-134-VI Topotecan
Topo I
Chemotherapy
0.0099907
-0.8909 1.0405 0.1644 0.5440
0.071904
0.95834
MDA-MB-361 Luminespib
HSP90
Misc
0.0071417
-0.8855 0.9781 0.3455 4.9987
0.0087421
0.9995
MDA-MB-134-VI INK-128
mTORC1/2
PI3K/mTOR
0.0033793
-0.8853 1.2003 0.2512 1.2527
0.007425
0.99747
HCC70 Ceritinib
ALK
RTK
3.1923
-0.8808 0.1379 0.0703 5.0000
3.9213
0.99483
MDA-MB-134-VI ABT-737
Bcl2/XL
Misc
1.7727
-0.8735 0.2629 0.1112 1.9770
3.09
0.99496
HCC1428 Ceritinib
ALK
RTK
1.2414
-0.8673 0.3014 0.1288 1.6178
2.4481
0.99584
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