Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
A-375 Vemurafenib AGK2 1.0000 0.5333
uM
48
hr
1 2049 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 263.62 NGFR rabbit IgG(H+L) / donkey NGFR 162.71
A375-B1-rep1
D5
COLO 858 Vemurafenib AGK2 0.3160 2.6667
uM
48
hr
1 564 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 311.41 NGFR rabbit IgG(H+L) / donkey NGFR 108.97
Colo858-A2-rep1
D5
WM-115 Vemurafenib AGK2 1.0000 0.5333
uM
48
hr
1 915 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 145.02 NGFR rabbit IgG(H+L) / donkey NGFR 1130.32
WM115-B1-rep1
D5
WM-115 Vemurafenib AGK2 1.0000 0.1067
uM
48
hr
2 1468 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.46 NGFR rabbit IgG(H+L) / donkey NGFR 1223.13
WM115-B2-rep2
D5
WM-115 Vemurafenib AGK2 1.0000 0.5333
uM
48
hr
2 1023 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 128.12 NGFR rabbit IgG(H+L) / donkey NGFR 1175.15
WM115-B1-rep2
D5
COLO 858 Vemurafenib AGK2 0.3160 2.6667
uM
48
hr
2 635 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 266.45 NGFR rabbit IgG(H+L) / donkey NGFR 71.47
Colo858-A2-rep2
D5
WM-115 Vemurafenib AGK2 1.0000 2.6667
uM
48
hr
2 313 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 133.37 NGFR rabbit IgG(H+L) / donkey NGFR 888.19
WM115-A2-rep2
D5
A-375 Vemurafenib AGK2 1.0000 0.1067
uM
48
hr
2 3264 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 185.18 NGFR rabbit IgG(H+L) / donkey NGFR 175.19
A375-B2-rep2
D5
COLO 858 Vemurafenib AGK2 0.3160 0.5333
uM
48
hr
2 1820 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 307.04 NGFR rabbit IgG(H+L) / donkey NGFR 114.96
Colo858-B1-rep2
D5
WM-115 Vemurafenib AGK2 1.0000 0.1067
uM
48
hr
1 1420 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 139.59 NGFR rabbit IgG(H+L) / donkey NGFR 1264.14
WM115-B2-rep1
D5
COLO 858 Vemurafenib AGK2 0.3160 0.5333
uM
48
hr
1 1897 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 317.36 NGFR rabbit IgG(H+L) / donkey NGFR 134.31
Colo858-B1-rep1
D5
A-375 Vemurafenib AGK2 1.0000 2.6667
uM
48
hr
2 1329 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 425.48 NGFR rabbit IgG(H+L) / donkey NGFR 176.32
A375-A2-rep2
D5
A-375 Vemurafenib AGK2 1.0000 0.1067
uM
48
hr
1 3383 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 234.29 NGFR rabbit IgG(H+L) / donkey NGFR 181.56
A375-B2-rep1
D5
COLO 858 Vemurafenib AGK2 0.3160 0.1067
uM
48
hr
1 2399 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 279.22 NGFR rabbit IgG(H+L) / donkey NGFR 124.75
Colo858-B2-rep1
D5
COLO 858 Vemurafenib AGK2 0.3160 0.1067
uM
48
hr
2 2858 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 305.97 NGFR rabbit IgG(H+L) / donkey NGFR 137.70
Colo858-B2-rep2
D5
WM-115 Vemurafenib AGK2 1.0000 2.6667
uM
48
hr
1 193 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 140.10 NGFR rabbit IgG(H+L) / donkey NGFR 876.79
WM115-A2-rep1
D5
A-375 Vemurafenib AGK2 1.0000 0.5333
uM
48
hr
2 1946 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 233.50 NGFR rabbit IgG(H+L) / donkey NGFR 153.50
A375-B1-rep2
D5
A-375 Vemurafenib AGK2 1.0000 2.6667
uM
48
hr
1 678 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 394.51 NGFR rabbit IgG(H+L) / donkey NGFR 132.96
A375-A2-rep1
D5
A-375 Vemurafenib Anacardic acid 1.0000 2.6667
uM
48
hr
2 1845 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 197.52 NGFR rabbit IgG(H+L) / donkey NGFR 193.43
A375-A2-rep2
G3
COLO 858 Vemurafenib Anacardic acid 0.3160 0.1067
uM
48
hr
2 1570 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 344.62 NGFR rabbit IgG(H+L) / donkey NGFR 122.24
Colo858-B2-rep2
G3
COLO 858 Vemurafenib Anacardic acid 0.3160 0.1067
uM
48
hr
1 1144 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 317.68 NGFR rabbit IgG(H+L) / donkey NGFR 153.35
Colo858-B2-rep1
G3
COLO 858 Vemurafenib Anacardic acid 0.3160 2.6667
uM
48
hr
2 998 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 267.99 NGFR rabbit IgG(H+L) / donkey NGFR 163.66
Colo858-A2-rep2
G3
A-375 Vemurafenib Anacardic acid 1.0000 0.5333
uM
48
hr
2 1745 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 183.73 NGFR rabbit IgG(H+L) / donkey NGFR 158.90
A375-B1-rep2
G3
COLO 858 Vemurafenib Anacardic acid 0.3160 0.5333
uM
48
hr
1 1751 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 322.89 NGFR rabbit IgG(H+L) / donkey NGFR 153.60
Colo858-B1-rep1
G3
A-375 Vemurafenib Anacardic acid 1.0000 0.1067
uM
48
hr
2 2049 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 170.49 NGFR rabbit IgG(H+L) / donkey NGFR 140.28
A375-B2-rep2
G3
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