Phosphorylation state and protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with combinations of two compounds (immunofluorescence dataset 1 of 4) - Dataset (ID:20274)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (568) Secondary Antibody (568) Protein Detected (568) Mean Fluorescence Intensity (568) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
A-375 Vemurafenib AZD8055 0.000 0.200
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1689.11 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 371.16 NGFR rabbit IgG(H+L) / donkey NGFR 370.45
A375-P7
E6
A-375 Vemurafenib AZD8055 1.000 0.200
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 953.39 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 203.29 NGFR rabbit IgG(H+L) / donkey NGFR 530.58
A375-P7
G6
A-375 Vemurafenib AZD8055 0.000 0.600
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1255.45 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 286.02 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 186.22
A375-P10
E7
A-375 Vemurafenib AZD8055 1.000 0.600
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 684.78 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 167.37 NGFR rabbit IgG(H+L) / donkey NGFR 532.87
A375-P7
D7
A-375 Vemurafenib AZD8055 0.316 0.200
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1065.67 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 221.73 NGFR rabbit IgG(H+L) / donkey NGFR 534.00
A375-P7
F6
A-375 Vemurafenib AZD8055 0.316 0.600
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 989.80 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 212.12 NGFR rabbit IgG(H+L) / donkey NGFR 424.21
A375-P7
F7
A-375 Vemurafenib AZD8055 1.000 0.600
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 695.94 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 192.03 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 280.62
A375-P10
D7
A-375 Vemurafenib AZD8055 1.000 0.600
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 784.40 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 188.16 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 239.79
A375-P10
G7
A-375 Vemurafenib AZD8055 0.000 0.600
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1583.62 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 345.10 NGFR rabbit IgG(H+L) / donkey NGFR 297.21
A375-P7
B7
A-375 Vemurafenib AZD8055 1.000 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 745.76 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 173.12 NGFR rabbit IgG(H+L) / donkey NGFR 644.03
A375-P7
D6
A-375 Vemurafenib AZD8055 0.000 0.600
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1607.03 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 317.34 NGFR rabbit IgG(H+L) / donkey NGFR 319.81
A375-P7
E7
A-375 Vemurafenib AZD8055 1.000 0.200
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 809.04 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 194.24 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 290.26
A375-P10
G6
A-375 Vemurafenib AZD8055 0.316 0.600
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 847.30 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 216.14 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 262.95
A375-P10
F7
A-375 Vemurafenib AZD8055 0.316 0.200
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 774.02 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 199.06 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 258.33
A375-P10
F6
A-375 Vemurafenib AZD8055 0.000 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1461.59 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 333.92 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 205.97
A375-P10
B6
A-375 Vemurafenib AZD8055 0.316 0.600
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 737.85 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 204.50 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 267.04
A375-P10
C7
A-375 Vemurafenib AZD8055 0.316 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 892.27 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 227.01 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 314.05
A375-P10
C6
A-375 Vemurafenib AZD8055 0.000 0.600
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1214.84 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 269.03 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 176.94
A375-P10
B7
A-375 Vemurafenib AZD8055 1.000 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 534.00 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 177.96 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 299.97
A375-P10
D6
A-375 Vemurafenib AZD8055 0.000 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1911.21 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 394.21 NGFR rabbit IgG(H+L) / donkey NGFR 310.04
A375-P7
B6
A-375 Vemurafenib AZD8055 0.316 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1015.43 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 227.72 NGFR rabbit IgG(H+L) / donkey NGFR 506.01
A375-P7
C6
A-375 Vemurafenib AZD8055 0.316 0.600
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 979.73 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 221.80 NGFR rabbit IgG(H+L) / donkey NGFR 400.84
A375-P7
C7
A-375 Vemurafenib AZD8055 0.000 0.200
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1301.07 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 298.21 c-Jun (pS73) rabbit IgG(H+L) / donkey c-Jun (pS73) 167.81
A375-P10
E6
A-375 Vemurafenib AZD8055 0.000 0.200
uM
48
hr
1 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 1464.57 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 324.97 S6 (pS240; pS244) rabbit IgG(H+L) / donkey S6 (pS240; pS244) 974.92
A375-P8
B6
A-375 Vemurafenib AZD8055 1.000 0.600
uM
48
hr
2 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 987.57 Rb (pS807; pS811) goat IgG(H+L) Rb (pS807; pS811) 184.95 NGFR rabbit IgG(H+L) / donkey NGFR 465.50
A375-P7
G7
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