Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 2 of 4: Calculated dose-response metrics. - Dataset (ID:20269)

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Cell Clinical Subtype Transcriptional Subtype Small Molecule Antibody Perturbagen Target Perturbagen Class Biological Replicate ID Conc Unit GR50 GEC50 GRmax GRinf GR Hill Coefficient GR_AOC GR r2 Nominal Division Rate
21MT-1
HER2amp
-
Z-Leu-Leu-Norvalinal
Proteasome
Proteasome
14191.189
uM
0.40746
0.57483
-0.6146 -0.6271 2.3620 0.6103
0.9968
2.9704
21NT
HER2amp
-
MG-132
Proteasome
Proteasome
14194.189
uM
0.10310
0.10891
-0.3512 -0.1578 5.0000 0.6651
0.5943
2.3616
21MT-1
HER2amp
-
MG-132
Proteasome
Proteasome
14191.189
uM
inf
inf
-0.1161 -0.1161 0.0000 0.5482
0.5418
2.9704
21MT-1
HER2amp
-
Z-Leu-Leu-Norvalinal
Proteasome
Proteasome
14607.189
uM
0.44295
0.66473
-0.8717 -0.8791 2.4993 0.7149
0.9937
1.3733
21NT
HER2amp
-
Disulfiram
Proteasome
Proteasome
13575.174
uM
25.85920
36.60680
-0.6014 -0.8791 2.9191 0.1524
0.9863
1.5845
21NT
HER2amp
-
MG-132
Proteasome
Proteasome
14194.189
uM
0.10310
0.10891
-0.3512 -0.1578 5.0000 0.6651
0.5943
2.3616
21MT-1
HER2amp
-
Dichloroacetate
PDK
PDK
13719.176
uM
inf
inf
0.9233 0.9233 0.0000 0.0596
-0.2426
0.8672
21MT-1
HER2amp
-
Methylglyoxal
13719.184
uM
680.32080
999.99990
-0.9954 -0.9645 2.7899 0.6345
0.9961
0.7600
21MT-1
HER2amp
-
MG-132
Proteasome
Proteasome
14607.189
uM
0.09589
0.20341
-0.9029 -0.9017 1.3707 0.8886
0.9922
1.3733
21MT-1
HER2amp
-
Torkinib
15382.211
uM
0.01093
0.03899
-0.2640 -0.3399 0.4078 0.7366
0.9935
1.1714
21NT
HER2amp
-
Bortezomib
Proteasome
Proteasome
14783.203
uM
3.0610
4.70130
-0.8093 -0.8292 2.2786 0.4078
0.9883
1.8667
21NT
HER2amp
-
Dichloroacetate
PDK
PDK
13575.176
uM
7.46330
16.77450
0.7977 -0.9991 1.3558 0.0319
0.6506
1.4733
21NT
HER2amp
-
Mebendazole
13575.174
uM
0.70544
0.60467
0.2760 0.2687 5.0000 0.2944
0.9408
1.5845
21NT
HER2amp
-
Methylglyoxal
13653.184
uM
371.60
1000.00000
-0.9322 -0.8591 1.0101 0.5941
0.9376
1.5871
21MT-1
HER2amp
-
Bortezomib
Proteasome
Proteasome
14779.203
uM
2.22370
3.73670
-0.7373 -0.7957 1.8347 0.4364
0.9894
1.9695
21MT-1
HER2amp
-
Bortezomib
Proteasome
Proteasome
14779.203
uM
2.22370
3.73670
-0.7373 -0.7957 1.8347 0.4364
0.9894
1.9695
21MT-1
HER2amp
-
Disulfiram
Proteasome
Proteasome
13719.174
uM
inf
0.02944
0.8637 0.8697 4.9974 0.0852
0.6419
0.8124
21MT-1
HER2amp
-
Mebendazole
13719.174
uM
31.97060
77.55140
0.0875 -1.0000 1.2398 0.1610
0.8782
0.8124
21MT-1
HER2amp
-
MG-132
Proteasome
Proteasome
14191.189
uM
inf
inf
-0.1161 -0.1161 0.0000 0.5482
0.5418
2.9704
21MT-1
HER2amp
-
MG-132
Proteasome
Proteasome
14607.189
uM
0.09589
0.20341
-0.9029 -0.9017 1.3707 0.8886
0.9922
1.3733
21MT-1
HER2amp
-
Nelfinavir
13719.174
uM
10.30820
13.49270
-0.9513 -1.0000 4.0808 0.1693
0.9959
0.8124
21MT-1
HER2amp
-
Ribavirin
15382.211
uM
inf
inf
0.9683 0.9683 0.0000 0.0416
0.0000
1.1714
21NT
HER2amp
-
Bortezomib
Proteasome
Proteasome
14783.203
uM
3.0610
4.70130
-0.8093 -0.8292 2.2786 0.4078
0.9883
1.8667
21NT
HER2amp
-
MG-132
Proteasome
Proteasome
14610.189
uM
0.09536
0.14625
-0.9556 -0.9536 2.4958 0.9558
0.9950
1.0787
21NT
HER2amp
-
MG-132
Proteasome
Proteasome
14610.189
uM
0.09536
0.14625
-0.9556 -0.9536 2.4958 0.9558
0.9950
1.0787
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