Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 2 of 4: Calculated dose-response metrics. - Dataset (ID:20269)

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Cell Clinical Subtype Transcriptional Subtype Small Molecule Antibody Perturbagen Target Perturbagen Class Biological Replicate ID Conc Unit GR50 GEC50 GRmax GRinf GR Hill Coefficient GR_AOC GR r2 Nominal Division Rate
BT-549
TNBC
Basal B
Gemcitabine
DNA replication
DNA replication
10261.131
uM
-inf
0.00002
-0.3245 -0.3912 0.1000 1.0766
0.7849
2.3992
BT-474
HER2amp
Luminal
Cetuximab
EGFR
ErbB
9163.026
uM
inf
0.00002
0.8122 0.8820 4.9564 0.0838
0.5768
0.3738
HCC70
TNBC
Basal A
Torkinib
15390.211
uM
-inf
0.00003
-0.9960 -0.9803 0.5245 1.8586
0.9905
0.5021
MDA-MB-468
TNBC
Basal A
Vinorelbine
TUBB
TUBB
7906.018
uM
0.00003
0.00009
-0.9241 -0.7076 0.8524 1.6148
0.7919
0.9087
ZR-75-1
HR+
Luminal
Torkinib
15346.211
uM
0.00002
0.00009
-0.6847 -0.6526 0.5569 1.5120
0.9820
0.6395
SUM1315MO2
TNBC
Basal B
Torkinib
15401.211
uM
-inf
0.00012
-0.9603 -0.8964 0.4331 1.6631
0.9588
0.4079
HCC3153
TNBC
Basal A
Ro 32-0432
PKC
PKC
10577.142
uM
inf
0.00015
0.8665 0.8748 5.0000 0.1168
0.5822
1.0584
MCF7
HR+
Luminal
Torkinib
15394.211
uM
0.00006
0.00015
-0.2414 -0.2040 0.3606 1.0163
0.9695
1.8299
HCC2185
TNBC
Luminal
Sirolimus
MTOR
MTOR
7463.068
uM
0.00019
0.00017
-0.0655 0.0169 0.3266 0.8520
0.8086
0.5887
HCC1954
HER2amp
Basal A
Vinorelbine
TUBB
TUBB
7837.042
uM
0.00015
0.00026
-0.8248 -0.4139 1.1755 1.2659
0.6601
1.6916
SUM44PE
HER2amp
Luminal
Sirolimus
MTOR
MTOR
7538.068
uM
0.00014
0.00030
-0.2424 -0.1582 0.3753 1.0105
0.7167
0.8203
T47DKBLUC
Unknown
Unknown
Torkinib
15360.211
uM
0.00023
0.00037
-0.1763 -0.1097 0.4213 0.9138
0.9795
0.8772
BT-549
TNBC
Basal B
Vinorelbine
TUBB
TUBB
7803.042
uM
0.00050
0.00052
-0.5972 -0.0656 2.5414 0.9089
0.7256
2.8270
HMT-3522 S1
Unknown
Unknown
Trametinib
MEK
MAPK
10124.012
uM
0.00074
0.00053
0.2498 0.2658 2.3479 0.6006
0.9280
1.9565
SUM52PE
HR+
Luminal
Ixabepilone
TUBB
TUBB
7541.095
uM
0.00031
0.00056
-0.9787 -0.3061 0.7899 1.0595
0.6623
1.4542
UACC-812
HER2amp
Luminal
Torkinib
15404.211
uM
0.00005
0.00056
-0.8141 -0.8007 0.3960 1.4387
0.9967
0.5754
T47D
HR+
Luminal
Torkinib
15340.211
uM
0.00038
0.00069
-0.2049 -0.1299 0.3943 0.8877
0.9641
1.5685
HCC1954
HER2amp
Basal A
GSK461364
PLK1
PLK
7839.001
uM
0.00067
0.00070
-0.4867 -0.1112 5.0000 0.8932
0.8549
1.8919
MDA-MB-468
TNBC
Basal A
GSK461364
PLK1
PLK
7904.001
uM
0.00066
0.00071
-0.0087 -0.2074 5.0000 1.0124
0.6937
1.3917
HCC202
HER2amp
Luminal
GSK461364
PLK1
PLK
7841.001
uM
0.00065
0.00073
-0.7519 -0.1312 2.0815 0.9082
0.6730
0.5424
BT-483
HR+
Luminal
Sirolimus
MTOR
MTOR
5908.069
uM
0.00124
0.00074
0.1221 0.1875 0.9066 0.6615
0.9618
0.6014
AU565
HER2amp
Luminal
GSK461364
PLK1
PLK
9035.001
uM
0.00071
0.00076
0.2153 -0.1767 5.0000 0.9858
0.7915
2.4291
HCC1954
HER2amp
Basal A
Ixabepilone
TUBB
TUBB
7457.094
uM
0.00051
0.00078
-0.8956 -0.6816 2.0313 1.5901
0.9463
1.8462
EFM-192C
HER2amp
Luminal
Torkinib
15292.211
uM
0.00077
0.00081
-0.2486 -0.0154 0.7454 0.8411
0.8375
1.7715
HCC1419
HER2amp
Luminal
Trametinib
MEK
MAPK
7818.05
uM
6.20090
0.00082
0.3938 0.4924 0.4692 0.3679
0.6443
0.9274
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