BYL719 KINOMEscan - Dataset (ID:20263)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Alpelisib | PIK3CA(I800L) | 0.0 | 100 | nM |
| Alpelisib | PIK3CA(H1047L) | 0.0 | 100 | nM |
| Alpelisib | PIK3CA(E542K) | 0.0 | 1000 | nM |
| Alpelisib | PIK3CA(M1043I) | 0.0 | 100 | nM |
| Alpelisib | PIK3CA | 0.0 | 1000 | nM |
| Alpelisib | PIK3CA(Q546K) | 0.0 | 1000 | nM |
| Alpelisib | PIK3CA(I800L) | 0.0 | 1000 | nM |
| Alpelisib | PIK3CA(E545K) | 0.0 | 1000 | nM |
| Alpelisib | PIK3CA(H1047L) | 0.0 | 1000 | nM |
| Alpelisib | PIK3CB | 0.0 | 1000 | nM |
| Alpelisib | PIK3CA(E545A) | 0.1 | 1000 | nM |
| Alpelisib | PIK3CA(C420R) | 0.2 | 1000 | nM |
| Alpelisib | PIK3CA(H1047Y) | 0.2 | 100 | nM |
| Alpelisib | PIK3CG | 0.3 | 1000 | nM |
| Alpelisib | PIK3CA(E545K) | 0.8 | 100 | nM |
| Alpelisib | PIK3CA(E542K) | 1.4 | 100 | nM |
| Alpelisib | PIK3CA(E545A) | 1.5 | 100 | nM |
| Alpelisib | PIK3CA(C420R) | 1.6 | 100 | nM |
| Alpelisib | PIK3CA(Q546K) | 2.1 | 100 | nM |
| Alpelisib | PIK3CA(M1043I) | 2.5 | 1000 | nM |
| Alpelisib | ABL1(H396P)-phosphorylated | 2.9 | 1000 | nM |
| Alpelisib | PIK3CA | 4.0 | 100 | nM |
| Alpelisib | PIK4CB | 7.7 | 1000 | nM |
| Alpelisib | ABL1-phosphorylated | 10.0 | 1000 | nM |
| Alpelisib | PIK3CG | 12.0 | 100 | nM |