Sorafenib KINOMEscan-2 - Dataset (ID:20192)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Sorafenib | DDR1 | 1.5 | nM |
Sorafenib | HIPK4 | 3.3 | nM |
Sorafenib | FLT3(K663Q) | 4.5 | nM |
Sorafenib | MLTK | 6.3 | nM |
Sorafenib | DDR2 | 6.6 | nM |
Sorafenib | RET(M918T) | 7.4 | nM |
Sorafenib | FLT3(N841I) | 11.0 | nM |
Sorafenib | RET | 13.0 | nM |
Sorafenib | FLT3 | 13.0 | nM |
Sorafenib | KIT(V559D) | 16.0 | nM |
Sorafenib | FLT3(R834Q) | 17.0 | nM |
Sorafenib | KIT(V559D,T670I) | 18.0 | nM |
Sorafenib | KIT(A829P) | 20.0 | nM |
Sorafenib | RET(V804M) | 22.0 | nM |
Sorafenib | KIT(L576P) | 25.0 | nM |
Sorafenib | CSF1R | 28.0 | nM |
Sorafenib | KIT | 28.0 | nM |
Sorafenib | FLT3(D835H) | 30.0 | nM |
Sorafenib | VGFR1 | 31.0 | nM |
Sorafenib | PGFRB | 37.0 | nM |
Sorafenib | RET(V804L) | 39.0 | nM |
Sorafenib | ERK8 | 46.0 | nM |
Sorafenib | VGFR2 | 59.0 | nM |
Sorafenib | PGFRA | 62.0 | nM |
Sorafenib | TIE1 | 68.0 | nM |