Breast cell line dose response to target inhibition measured by high throughput microscopy - Dataset (ID:20136)

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Small Molecule Cell Line Drug Concentration Conc Units Timepoint Timepoint Units Measured pERK (Alexa 488) Measured p-Rb (Alexa 568) Alexa Fluor 647 Measured p-Akt/p-4EBP1/p-S6 (Alexa 647) Image
Dactolisib AU565
3.16
nM
24
hr
451.27 106.53
p-Akt
105.91 image if available
Dactolisib T47D
3.16
nM
6
hr
112.31 65.77
p-Akt
19.14 image if available
Dactolisib MCF 10A
1.0
nM
24
hr
332.80 131.47
p-Akt
43.15 image if available
Dactolisib AU565
3.16
nM
6
hr
259.31 60.60
p-Akt
24.45 image if available
Dactolisib MCF 10A
3.16
nM
6
hr
394.32 173.00
p-Akt
43.59 image if available
Dactolisib MCF 10A
3.16
nM
24
hr
306.83 142.69
p-Akt
34.75 image if available
Dactolisib HCC1954
1.0
nM
6
hr
151.35 38.59
p-Akt
20.04 image if available
Dactolisib MCF 10A
1.0
nM
6
hr
437.12 174.36
p-Akt
52.90 image if available
Dactolisib T47D
1.0
nM
6
hr
90.24 35.16
p-Akt
13.70 image if available
Dactolisib T47D
1.0
nM
24
hr
138.24 90.29
p-Akt
47.16 image if available
Dactolisib HCC1954
3.16
nM
6
hr
218.96 75.61
p-Akt
41.58 image if available
Dactolisib HCC1954
3.16
nM
24
hr
294.20 99.05
p-Akt
76.79 image if available
Dactolisib MCF 10A
0 (control)
24
hr
351.94 125.18
p-Akt
50.36 image if available
Dactolisib T47D
0 (control)
6
hr
99.23 26.75
p-Akt
14.05 image if available
Dactolisib AU565
1.0
nM
24
hr
494.41 109.15
p-Akt
109.06 image if available
Dactolisib HCC1954
1.0
nM
24
hr
302.85 101.27
p-Akt
76.62 image if available
Dactolisib MCF 10A
0 (control)
6
hr
436.72 165.98
p-Akt
55.27 image if available
Dactolisib T47D
0 (control)
24
hr
165.27 86.01
p-Akt
60.10 image if available
Dactolisib AU565
0 (control)
24
hr
496.14 121.03
p-Akt
137.91 image if available
Dactolisib AU565
1.0
nM
6
hr
217.79 50.25
p-Akt
22.45 image if available
Dactolisib AU565
0 (control)
6
hr
235.49 54.01
p-Akt
23.90 image if available
Dactolisib HCC1954
0 (control)
6
hr
262.96 93.99
p-Akt
56.53 image if available
Dactolisib HCC1954
0 (control)
24
hr
357.28 117.27
p-Akt
79.92 image if available
Dactolisib AU565
10.0
nM
6
hr
210.20 46.30
p-Akt
19.17 image if available
Dactolisib T47D
3.16
nM
24
hr
138.41 87.20
p-Akt
40.75 image if available
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  • 1 to 25 of 2880 records