Breast cell line dose response to target inhibition measured by high throughput microscopy - Dataset (ID:20136)

Filter results: >>>>
Small Molecule Cell Line Drug Concentration Conc Units Timepoint Timepoint Units Measured pERK (Alexa 488) Measured p-Rb (Alexa 568) Alexa Fluor 647 Measured p-Akt/p-4EBP1/p-S6 (Alexa 647) Image
Dactolisib AU565
100.0
nM
6
hr
290.65 59.15
p-Akt
17.08 image if available
Dactolisib AU565
100.0
nM
24
hr
377.63 60.16
p-Akt
25.52 image if available
Gefitinib HCC1954
100.0
nM
6
hr
166.09 41.51
p-Akt
23.50 image if available
Gefitinib HCC1954
100.0
nM
24
hr
271.49 112.65
p-Akt
74.36 image if available
Torkinib HCC1954
31.6
nM
6
hr
150.07 28.76
p-Akt
14.38 image if available
Torkinib HCC1954
31.6
nM
24
hr
250.65 86.99
p-Akt
39.42 image if available
GSK1059615 HCC1954
100.0
nM
6
hr
324.83 87.89
p-Akt
34.01 image if available
GSK1059615 HCC1954
100.0
nM
24
hr
285.12 84.64
p-Akt
37.56 image if available
MK2206 HCC1954
100.0
nM
6
hr
239.59 77.83
p-Akt
17.44 image if available
MK2206 HCC1954
100.0
nM
24
hr
248.97 102.29
p-Akt
31.95 image if available
Triciribine HCC1954
100.0
nM
6
hr
200.10 73.80
p-Akt
29.38 image if available
Triciribine HCC1954
100.0
nM
24
hr
238.17 94.17
p-Akt
36.41 image if available
Dactolisib HCC1954
100.0
nM
6
hr
186.97 55.42
p-Akt
16.95 image if available
Dactolisib HCC1954
100.0
nM
24
hr
240.30 68.59
p-Akt
21.56 image if available
Gefitinib MCF 10A
100.0
nM
6
hr
345.12 168.30
p-Akt
37.38 image if available
Gefitinib MCF 10A
100.0
nM
24
hr
258.63 122.31
p-Akt
28.67 image if available
Torkinib MCF 10A
31.6
nM
6
hr
436.07 147.11
p-Akt
29.06 image if available
Torkinib MCF 10A
31.6
nM
24
hr
400.54 150.17
p-Akt
24.66 image if available
GSK1059615 MCF 10A
100.0
nM
6
hr
316.39 158.33
p-Akt
27.50 image if available
GSK1059615 MCF 10A
100.0
nM
24
hr
326.44 133.59
p-Akt
27.72 image if available
MK2206 MCF 10A
100.0
nM
6
hr
358.46 151.32
p-Akt
25.55 image if available
MK2206 MCF 10A
100.0
nM
24
hr
301.03 149.65
p-Akt
23.12 image if available
Triciribine MCF 10A
100.0
nM
6
hr
360.87 152.35
p-Akt
25.66 image if available
Triciribine MCF 10A
100.0
nM
24
hr
231.53 128.71
p-Akt
20.57 image if available
Dactolisib MCF 10A
100.0
nM
6
hr
342.01 143.79
p-Akt
24.33 image if available