Metrics other than potency reveal systematic variation in responses to cancer drugs - Dataset (ID:20120)
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Small Molecule | Cell Line | log10[max. dose (M)] | R^2 (goodness of fit) | log10[EC50 (M)] | log10[IC50 (M)] | log10[GI50 (M)] | HillSlope | E_inf | E_max | AUC |
---|---|---|---|---|---|---|---|---|---|---|
Torkinib | MCF7 | -4.3010 | 0.9482 | -10.1570 | -9.6593 | -10.3750 | 0.4305 | 0.1950 | 0.1974 | 2.6031 |
Torkinib | ZR-75-1 | -4.3010 | 0.9479 | -9.8430 | -8.9499 | -10.7280 | 0.5030 | 0.3223 | 0.3234 | 3.6921 |
Torkinib | HCC70 | -4.3010 | 0.9415 | -9.6690 | -9.5655 | -12.1070 | 0.3058 | 0.0350 | 0.0565 | 2.0727 |
Torkinib | T47D | -4.3010 | 0.9460 | -9.4110 | -8.5983 | -9.5701 | 0.4377 | 0.2796 | 0.2838 | 3.7359 |
Torkinib | T47DKBLUC | -4.3010 | 0.9063 | -9.3870 | -5.1956 | -9.6065 | 0.4163 | 0.4910 | 0.4949 | 5.3140 |
Ixabepilone | MDA-MB-231 | -4.4045 | 0.9286 | -9.2455 | -9.2112 | -9.2591 | 1.4930 | 0.1324 | 0.1324 | 2.3981 |
GSK461364 | MDA-MB-157 | -4.4776 | 0.9444 | -9.0436 | -8.9391 | -9.0610 | 2.6360 | 0.2340 | 0.2340 | 3.5893 |
Torkinib | HCC38 | -4.3010 | 0.9596 | -8.9020 | -8.8385 | -9.6108 | 0.5908 | 0.0409 | 0.0428 | 2.3342 |
Docetaxel | SUM149PT | -5.0000 | 0.9360 | -8.8090 | -8.6657 | -8.8072 | 2.3100 | 0.2665 | 0.2665 | 4.7876 |
Docetaxel | SUM159PT | -5.0000 | 0.9753 | -8.7915 | -8.7477 | -8.8094 | 2.1380 | 0.0956 | 0.0956 | 3.6627 |
Torkinib | UACC-812 | -4.3010 | 0.9736 | -8.7280 | -7.8546 | -10.2600 | 0.3573 | 0.2563 | 0.2753 | 4.2197 |
Torkinib | MCF 10F | -4.3010 | 0.9683 | -8.7050 | -8.2104 | -8.8465 | 0.5975 | 0.2470 | 0.2488 | 3.9764 |
Ixabepilone | Hs 578T | -4.4045 | 0.9537 | -8.6775 | -8.6117 | -8.7153 | 1.3270 | 0.1267 | 0.1267 | 3.5228 |
Docetaxel | SUM52PE | -5.0000 | 0.9765 | -8.6740 | -8.4669 | -8.7954 | 1.5570 | 0.2588 | 0.2588 | 4.8421 |
Trametinib | HCC1806 | -4.7773 | 0.8477 | -8.6718 | -4.7773 | -6.3239 | 2.3950 | 0.6729 | 0.6729 | 7.0514 |
Omipalisib | 184A1 | -4.4776 | 0.9136 | -8.6666 | -8.1611 | -8.7804 | 0.9289 | 0.3302 | 0.3303 | 4.7168 |
Docetaxel | 184B5 | -5.0000 | 0.8431 | -8.6610 | -5.0000 | -8.3663 | 2.1670 | 0.6800 | 0.6800 | 7.7232 |
Docetaxel | MCF 10F | -5.0000 | 0.9663 | -8.6590 | -8.4334 | -8.6146 | 1.7160 | 0.2946 | 0.2946 | 4.9801 |
Gemcitabine | HCC1806 | -3.8416 | 0.9790 | -8.6516 | -8.5897 | -8.7366 | 2.1030 | 0.1252 | 0.1252 | 2.5814 |
Docetaxel | MCF 10A | -5.0000 | 0.9724 | -8.6485 | -8.4958 | -8.6453 | 1.4580 | 0.1865 | 0.1866 | 4.3758 |
Docetaxel | HCC1954 | -5.0000 | 0.9115 | -8.6430 | -8.5724 | -8.8092 | 1.2620 | 0.0624 | 0.0624 | 3.8091 |
Docetaxel | Hs 578T | -5.0000 | 0.9693 | -8.6405 | -8.5044 | -8.8125 | 1.4793 | 0.1759 | 0.1761 | 4.2545 |
Docetaxel | MCF12A | -5.0000 | 0.9298 | -8.6260 | -8.2368 | -8.6178 | 1.3250 | 0.3435 | 0.3436 | 5.1394 |
GSK461364 | HCC1954 | -4.4776 | 0.9031 | -8.6121 | -8.5601 | -8.6498 | 3.7270 | 0.1966 | 0.1966 | 3.8376 |
Docetaxel | HCC38 | -5.0000 | 0.9818 | -8.6120 | -8.4709 | -8.7384 | 1.9535 | 0.2238 | 0.2238 | 4.5902 |