XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
70.4
10
uM
XMD-12 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
87.9
10
uM
XMD-12 PC-3 AGK
ATVFLNPAACkGK
ATP
-6.7
10
uM
XMD-12 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
88.8
10
uM
XMD-12 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
91.5
10
uM
XMD-12 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
88.7
10
uM
XMD-12 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
90.3
10
uM
XMD-12 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
-7.0
10
uM
XMD-12 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
1.1
10
uM
XMD-12 PC-3 ATR
FYIMMCkPK
ATP
16.8
10
uM
XMD-12 HeLa ATR
FYIMMCkPK
ATP
-2.1
10
uM
XMD-12 HeLa AurB
SHFIVALkVLFK
Lys1
95.0
10
uM
XMD-12 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
-4.3
10
uM
XMD-12 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
-6.9
10
uM
XMD-12 HeLa BTK
GQYDVAIkMIK
Lys1
28.3
10
uM
XMD-12 HeLa CaMK1a
LVAIkCIAK
Lys1
-16.8
10
uM
XMD-12 HeLa CAMK1D
LFAVkCIPK
Lys1
-29.5
10
uM
XMD-12 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
23.5
10
uM
XMD-12 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
33.0
10
uM
XMD-12 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
19.3
10
uM
XMD-12 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
22.4
10
uM
XMD-12 PC-3 CDK10
DLkVSNLLMTDK
Lys2
81.3
10
uM
XMD-12 PC-3 CDK11,CDK8
DLkPANILVMGEGPER
Lys2
7.1
10
uM
XMD-12 PC-3 CDK14
LVALkVIR
Lys1
1.1
10
uM
XMD-12 PC-3 CDK16
LTDNLVALkEIR
Lys1
-11.1
10
uM
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  • 1 to 25 of 241 records