XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 70.4 | 10 | uM |
XMD-12 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 87.9 | 10 | uM |
XMD-12 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -6.7 | 10 | uM |
XMD-12 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 88.8 | 10 | uM |
XMD-12 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 91.5 | 10 | uM |
XMD-12 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 88.7 | 10 | uM |
XMD-12 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 90.3 | 10 | uM |
XMD-12 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -7.0 | 10 | uM |
XMD-12 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 1.1 | 10 | uM |
XMD-12 | PC-3 | ATR | FYIMMCkPK | ATP | 16.8 | 10 | uM |
XMD-12 | HeLa | ATR | FYIMMCkPK | ATP | -2.1 | 10 | uM |
XMD-12 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 95.0 | 10 | uM |
XMD-12 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | -4.3 | 10 | uM |
XMD-12 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -6.9 | 10 | uM |
XMD-12 | HeLa | BTK | GQYDVAIkMIK | Lys1 | 28.3 | 10 | uM |
XMD-12 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -16.8 | 10 | uM |
XMD-12 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -29.5 | 10 | uM |
XMD-12 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 23.5 | 10 | uM |
XMD-12 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 33.0 | 10 | uM |
XMD-12 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.3 | 10 | uM |
XMD-12 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 22.4 | 10 | uM |
XMD-12 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 81.3 | 10 | uM |
XMD-12 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 7.1 | 10 | uM |
XMD-12 | PC-3 | CDK14 | LVALkVIR | Lys1 | 1.1 | 10 | uM |
XMD-12 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -11.1 | 10 | uM |