XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
46.7
10
uM
XMD-12 HeLa SYK
ISDFGLSkALR
Activation Loop
2.1
10
uM
XMD-12 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
-12.6
10
uM
XMD-12 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-24.0
10
uM
XMD-12 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-7.6
10
uM
XMD-12 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
27.4
10
uM
XMD-12 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-23.4
10
uM
XMD-12 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
51.7
10
uM
XMD-12 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-26.4
10
uM
XMD-12 PC-3 NEK9
LGDYGLAkK
Activation Loop
3.4
10
uM
XMD-12 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-21.4
10
uM
XMD-12 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
27.3
10
uM
XMD-12 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
12.8
10
uM
XMD-12 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
50.3
10
uM
XMD-12 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
70.4
10
uM
XMD-12 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-14.1
10
uM
XMD-12 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
10
uM
XMD-12 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-11.9
10
uM
XMD-12 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
3.9
10
uM
XMD-12 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
70.5
10
uM
XMD-12 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
2.2
10
uM
XMD-12 HeLa NEK9
LGDYGLAkK
Activation Loop
-5.2
10
uM
XMD-12 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
61.2
10
uM
XMD-12 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
11.2
10
uM
XMD-12 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
26.6
10
uM
  • Page 1 of 10
  • 1 to 25 of 241 records