XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD-12 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 46.7 | 10 | uM |
XMD-12 | HeLa | SYK | ISDFGLSkALR | Activation Loop | 2.1 | 10 | uM |
XMD-12 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | -12.6 | 10 | uM |
XMD-12 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -24.0 | 10 | uM |
XMD-12 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -7.6 | 10 | uM |
XMD-12 | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | 27.4 | 10 | uM |
XMD-12 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -23.4 | 10 | uM |
XMD-12 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 51.7 | 10 | uM |
XMD-12 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | -26.4 | 10 | uM |
XMD-12 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 3.4 | 10 | uM |
XMD-12 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -21.4 | 10 | uM |
XMD-12 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 27.3 | 10 | uM |
XMD-12 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | 12.8 | 10 | uM |
XMD-12 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | 50.3 | 10 | uM |
XMD-12 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 70.4 | 10 | uM |
XMD-12 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -14.1 | 10 | uM |
XMD-12 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 10 | uM | |
XMD-12 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -11.9 | 10 | uM |
XMD-12 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | 3.9 | 10 | uM |
XMD-12 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 70.5 | 10 | uM |
XMD-12 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 2.2 | 10 | uM |
XMD-12 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -5.2 | 10 | uM |
XMD-12 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | 61.2 | 10 | uM |
XMD-12 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | 11.2 | 10 | uM |
XMD-12 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 26.6 | 10 | uM |