CP466722 KINOMEscan - Dataset (ID:20028)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
CP466722 | ABL1(H396P)-nonphosphorylated | 0.0 | 10 | uM |
CP466722 | ABL1(Q252H)-nonphosphorylated | 0.0 | 10 | uM |
CP466722 | TYK2(JH2domain-pseudokinase) | 0.0 | 10 | uM |
CP466722 | HIPK3 | 0.0 | 10 | uM |
CP466722 | DYRK1A | 0.1 | 10 | uM |
CP466722 | ABL1(F317L)-phosphorylated | 0.1 | 10 | uM |
CP466722 | KIT(D816V) | 0.2 | 10 | uM |
CP466722 | PLK4 | 0.2 | 10 | uM |
CP466722 | ABL1(H396P)-phosphorylated | 0.2 | 10 | uM |
CP466722 | NEK6 | 0.2 | 10 | uM |
CP466722 | ABL1(Q252H)-phosphorylated | 0.2 | 10 | uM |
CP466722 | ACVR1 | 0.2 | 10 | uM |
CP466722 | ABL1(Y253F)-phosphorylated | 0.3 | 10 | uM |
CP466722 | DYRK2 | 0.3 | 10 | uM |
CP466722 | CDKL5 | 0.3 | 10 | uM |
CP466722 | ABL1-phosphorylated | 0.3 | 10 | uM |
CP466722 | BMPR1B | 0.3 | 10 | uM |
CP466722 | FLT3(N841I) | 0.4 | 10 | uM |
CP466722 | AURKB | 0.4 | 10 | uM |
CP466722 | PIK3C2B | 0.4 | 10 | uM |
CP466722 | ABL1(E255K)-phosphorylated | 0.4 | 10 | uM |
CP466722 | JAK1(JH2domain-pseudokinase) | 0.4 | 10 | uM |
CP466722 | YSK4 | 0.5 | 10 | uM |
CP466722 | RPS6KA4(Kin.Dom.2-C-terminal) | 0.6 | 10 | uM |
CP466722 | ERK8 | 0.6 | 10 | uM |